Meriana Steroid Exemestane Aromasin Bakeng sa Antitumor CAS
CAS: | 107868-30-4 | Lehlalosi: | Aromasin; Exemestan |
---|---|---|---|
MF: | C20H24O2 | MW: | 296.4 |
Ponahalo: | Phofo e tšoeu ea Letlalo | Sebelisa: | E sebelisetsoa ho loants'a mofetše oa matsoele |
Meriana Steroid Exemestane Aromasin Bakeng sa Antitumor CAS 107868-30-4
Qaqileng e potlakileng
Lebitso la Sehlahisoa |
Seemahale
|
Lehlalosi |
Aromasin; Exemestan; Exemestane
|
CAS |
107868-30-4
|
MF |
C20H24O2
|
MW |
296.4
|
Qhibiliha Point |
155.13 ° C
|
Ho qhibiliha |
DMSO: ≥20mg / mL
|
Ponahalo |
Phofo e tšoeu ea kristale
|
E tloaelehileng |
Khoebo e Tloaelehileng
|
Tšebeliso |
Aromasin e sebelisetsoa ho loantša mofets'e oa matsoele le ho phahamisa testosterone 'meleng
|
Tlhaloso
Exemestane ke aromatase inhibitor. Sena se bolela hore e thibela enzyme aromatase (e fumanoang mesifa ea 'mele, letlalo, letsoele le mafura), e sebelisetsoang ho fetola li-androgens (lihormone tse hlahisoang ke litšoelesa tsa adrenal) ho ba estrogen. Ha ho se na estrogen, lihlahala tse itšetlehileng ka hormone ena bakeng sa kholo li tla fokotseha.
Exemestanes Aromasin ke ntho e ke keng ea fetoha, steroidal aromatase inactivator, e amanang hantle le karolo ea tlhaho ea androstenedione. E sebetsa joalo ka karoloana ea bohata bakeng sa enzyme ea aromatase, 'me e sebetsoa ho ba lipakeng tse tlamang se sa fetoheng sebakeng sa enzyme se bakang ho se sebetse, phello e tsejoang hape e le "thibelo ea ho ipolaea." Ka ho ts'oana ka mokhoa o ts'oanang le sepheo sa enzyme, Exemestanes Aromasin e tlama ka ho sa feleng ho li-enzyme, ho li thibela ho fetola androgen ho estrogen.
Kopo
Aromasin e sebelisetsoa ho loantša mofets'e oa matsoele le ho phahamisa testosterone 'meleng. Exemestane e thibela ts'ebetso ea monko o monate. Kahoo e theola bongata ba estrogen 'meleng. Kankere ea matsoele ea pele, ho nka exemestane ho ka thusa ho emisa mofetše oa matsoele ho khutla. Kankere ea matsoele e tsoetseng pele lisele tsa mofetše li ka hola butle hanyane kapa tsa emisa ho hola ka botlalo.
Exemestane (Aromasin) ke sethethefatsi se sebelisetsoang ho alafa mofetše oa matsoele. Ke setho sa sehlopha sa lithethefatsi tse tsejoang e le aromatase inhibitors. Mefuta e meng ea mofetše oa matsoele e hloka estrogen ho hola. Kankere eo e na le li-receptor tsa estrogen (ER), 'me e bitsoa ER-positive. Ba kanna ba bitsoa estrogen-reaction, hormonally-response, kapa hormone-receptor-positive. Aromatase ke enzyme e kopanyang estrogen. Aromatase inhibitors e thibela synthesis ea estrogen. Sena se theola boemo ba estrogen, mme se liehisa kholo ea mofetše.
Ga tlhaloso
Ntho | Ga tlhaloso |
Sephetho
|
Tlhaloso | Phofo e tšoeu ea Letlalo |
Phofo e Tšoeu
|
Boitsebiso | E ntle |
E ntle
|
Thlahlobo (ke HPLC) | 98.0 ~ 102.0% |
98.64%
|
Ho monya (E1cm) | 465 ~ 495 |
EA-482.5
|
Qhibiliha Point | 191 ~ 195 ° C |
193.5 ~ 195.0 ° C
|
Tahlehelo Ka Omisa | 0.5%, max |
0.19%
|
Itseng chenchana | + 288 ° ~ + 298 ° |
+ 290.2 °
|
Masalla On thothetsang molelo | 0,1%, max |
0.03%
|
Lintho tse amanang | Kakaretso: 1.5% max |
<1.3%
|
Masoha: 0.5%, max |
<0.4%
|
|
Masalla a Solvents | 0,2%, max |
0,0%
|
Lisebelisoa tse boima | Boholo ba 20PPm |
<10PPm
|
Tekanyo
Sena se ipapisitse le motho ka mong, hape, le bongata ba metsoako e monko o monate eo motho eo a e sebelisang. Ka kakaretso, tekanyetso e ntle ea ho qala ke 12.5mg ED (letsatsi le leng le le leng) kapa 25mg EOD (letsatsi le leng le le leng). Mosebelisi o tlameha ho sebelisa mosebetsi oa mali ho bona hore na 'mele ea bona e sebetsana joang le litekanyetso tseo a li khethang ebe o ikamahanya le moo ho hlokahalang. Basebelisi ba nang le boiphihlelo ba anabolic steroid hangata ba tla fumana tekanyetso eo ba e ratang mme ba e khomarele ntle le mathata. Joalokaha ke se ke boletse, haeba u qala ho hlokomela mathata a kopaneng joale lethal dose le lokela ho theoloa; ka lehlakoreng le leng, haeba u qala ho hlokomela mahlakore afe kapa afe a amanang le estrogen, joalo ka boikhohomoso kapa matsoele a thata kapa ho boloka metsi, ke nako ea ho eketsa litekanyetso.
Lihlahisoa tse ling tse chesang tse rekisoang:
Lebitso la Sehlahisoa | CAS Che. | ||
Letoto la Testosterone | |||
Enanthate ea Testosterone | CAS 315-37-7 | ||
Motheo oa Testosterone | CAS 58-22-0 | ||
Testosterone Acetate | CAS 1045-69-8 | ||
Testosterone Propionate | CAS 57-85-2 | ||
Testosterone Cypionate | CAS 58-20-8 | ||
Testosterone phenylpropionate | CAS 1255-49-8 | ||
Testosterone Isocaproate | CAS 15262-86-9 | ||
Testosterone Decanoate | CAS 5721-91-5 | ||
Testosterone Sustanon 250 | / | ||
Testosterone e sa tsitsang | CAS 5949-44-0 | ||
Fluoxymesterone (Halotestin) | CAS 76-43-7 | ||
17-Methyltestosterone | CAS 58-18-4 | ||
Mestanolone | CAS 521-11-9 | ||
Mesterolone (Proviron) | CAS 1424-00-6 | ||
Molomo Turinabol | CAS 2446-23-3 | ||
17a-Methyl-1-testosterone | CAS 65-04-3 | ||
Clostebol acetate (Turinabol) | CAS 855-19-6 | ||
1-Testosterone Cypiontae | CAS 1965-6-5 | ||
Letoto la Nandrolone | |||
Nandrolone | CAS 434-22-0 | ||
Nandrolone Decanoate (DECA) | CAS 360-70-3 | ||
Nandrolone Phenypropionate (Durabolin) | CAS 62-90-8 | ||
Metsoalle ea Stanolone (Androstanolone) | CAS 521-18-6 | ||
Mibolerone | CAS 3704-09-4 | ||
Nandrolone Propionbate | CAS | ||
Nandrolone Cypionate | CAS 601-63-8 | ||
Letoto la Trenbolone | |||
Trenbolone Acetate (Finaplix H / Revalor-H) | CAS 10161-34-9 | ||
Enanthate ea Trenbolone | CAS 10161-33-8 | ||
Metribolone (Methyltrienolone) | CAS 965-93-5 | ||
Trenbolone Hexahydrobenzyl Carbonate (parabolan) | CAS 23454-33-3 | ||
Motheo oa Trenbolone | CAS 10161-33-8 | ||
Tibolone | CAS 5630-53-5 | ||
Letoto la Boldenone | |||
Boldenone Base | CAS 846-48-0 | ||
Boldenone Undecylenate (Equipoise) | CAS 13103-34-9 | ||
Boldenone ea acetate | CAS 2363-59-9 | ||
Boldenone Cypionate | CAS 106505-90-2 | ||
Li-steroids tsa molomo | |||
Oxymetholone (Anadrol) | CAS 434-07-1 | ||
Oxandrolone (Anavar) | CAS 53-39-4 | ||
Stanozolol (Winstrol) | CAS 10418-03-8 | ||
Stanozolol (Winstrol) Phofo e Nyane | CAS 10418-03-8 | ||
Dianabol (Metandienone) | CAS 72-63-9 | ||
Letoto la Drostanolone | |||
Drostanolone Propionate (Masteron) | CAS 521-12-0 | ||
Enosthate ea Drostanolone | CAS 472-61-1 | ||
Methasterone (Superdrol) | CAS 3381-88-2 | ||
Letoto la Methenolone | |||
Enanthate ea Methenolone | CAS 303-42-4 | ||
Methenolone Acetate / Primobolan | CAS 434-05-9 | ||
Li-steroid tse khahlanong le Estrogen | |||
Tamoxifen | CAS 10540-29-1 | ||
Tamoxifen Citrate (Nolvadex) | CAS 54965-24-1 | ||
Clomiphene citrate | CAS 50-41-9 | ||
Toremifene citrate | CAS 89778-27-8 | ||
Exemestane (Aromasin) | CAS 107868-30-4 | ||
Formestane | CAS 566-48-3 | ||
Anastrozole (Arimidex) | CAS 120511-73-1 | ||
Letrazole (Femara) | CAS 112809-51-5 | ||
Ntlafatso ea thobalano | |||
Cialis (Tadalafil) | CAS 171596-29-5 | ||
Sildenafil Citrate (Viagra) | CAS 171599-83-0 | ||
Sildenafil Mesylate | / | ||
Vardenafil hydrochloride (Levitra) | CAS 224785-91-5 | ||
HCL | CAS 119356-77-3 | ||
Dutasteride (Avodart) | CAS 164656-23-9 | ||
Finasteride | CAS 98319-26-7 | ||
Yohimbine HCL | CAS 65-19-0 | ||
Motsoako oa li-steroid | |||
Benzyl Benzoate | CAS 120-51-4 | ||
Benzyl Joala | CAS 100-51-6 | ||
Oli ea Peo ea Morara | CAS 85594-37-2 | ||
Ethyl Oleate | CAS 111-62-6 | ||
Guaiakol | CAS 90-05-1 | ||
Polysorbate 80 (Mahareng a 80) | CAS 9005-65-6 | ||
Nhua polyethylene Glycol (mokotla) | CAS 25322-68-3 | ||
Propylene Glycol | CAS 57-55-6 | ||
Oli ea MCT | |||
Lihlooho tsa SARM | |||
MK-2866 (Ostarine, Enobosarm) | CAS 841205-47-8 | ||
GW501516 (GSK-516, Cardarine) | CAS 317318-70-0 | ||
MK-677 (Ibutamoren) | CAS 159634-47-6 | ||
S-4 (Andarine, GTX-007) | CAS401900-40-1 | ||
LGD-4033 | CAS1165910-22-4 | ||
SR9009 | CAS1379686-30-2 | ||
MOTSOALLE | CAS1379686-29-9 | ||
EA-11 | CAS431579-34-9 | ||
RAD140 | CAS1182367-47-0 | ||
AICAR (Acadesine) | CAS 2627-69-2 | ||
Li-hormone tsa polypeptide | |||
CJC1295 ntle le DAC | CAS 863288-34-0 | ||
CJC1295 le DAC | CAS 863288-34-0 | ||
Hexarelin | CAS 140703-51-1 | ||
MGF | |||
KHOTHATSO MGF | |||
EA-1-MT | CAS 75921-69-6 | ||
EA-2-MT | CAS 121062-08-6 | ||
GHRP-2 | CAS 158861-67-7 | ||
GHRP-6 | CAS 87616-84-0 | ||
Ipamorelin | CAS 170851-70-4 | ||
Sermorelin | CAS 86168-78-7 | ||
Oxytocin | CAS 50-56-6 | ||
TB500 | CAS 77591-33-4 | ||
Pentadecapeptide BPC 157 | |||
EA-9604 | CAS 221231-10-3 | ||
Litlhapi | CAS 57773-63-4 | ||
Tesamorelin | CAS 218949-48-5 |
Melemo:
Boleng 1.High le theko tlhōlisano:
(1) Tekanyetso: BP / USP
(2) Hloekileng Tsohle≥99%
(3) Re moetsi mme re ka fana ka lihlahisoa tsa boleng bo holimo ka theko ea fektheri.
Ho pepa ka potlako le ka polokeho
(1) Sephutheloana se ka romelloa ka mor'a lihora tse 24 ka mor'a ho lefa
(2) Ho romelloa ka mokhoa o sireletsehileng le o masene.Mekhoa e fapaneng ea lipalangoang eo u ka e khethang.
(3) Sekhahla sa ho feta sa Bolaoli ≥99%
(4) Re na le moemeli oa rona / remailer / distributor ea ka re thusang ho romella lihlahisoa tsa rona kapele haholo hape re bolokehile, 'me re na le setoko moo bakeng sa ho fetisa.
3.Re na le bareki lefatšeng ka bophara.
(1) Ts'ebeletso ea profeshenale le boiphihlelo bo ruileng li etsa hore bareki ba phutholohe, setoko se lekaneng le phano e potlakileng li fihlela takatso ea bona.
(2) Tlhaloso ea 'maraka le maikutlo a thepa li tla ananeloa, ho fihlela litlhoko tsa bareki ke boikarabello ba rona.
(3) Boleng bo phahameng, theko ea tlholisano, ho fana ka potlako, ts'ebeletso ea maemo a pele e fumana ts'epo le thoriso ho tsoa ho bareki.