99% Peptide Hormone Ipamorelin 2mg / Vial bakeng sa ho haha 'mele CAS 170851-70-4
CAS NO.: | 170851-70-4 | Limolek'hule Mokgwa wa ho Nahana: | 38H49N9O5 |
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Boima ba limolek'hule: | 711.853 | Thlahlobo: | 99.5% |
Ponahalo: | Phofo e tšoeu e tšoeu | Tšebeliso: | Ho haha 'mele |
Injectable Peptide Hormone Ipamorelin 2mg / Vial bakeng sa ho haha 'mele CAS 170851-70-4
Qaqileng e potlakileng
Lebitso la Sehlahisoa |
Ipamorelin
|
Mabitso |
696: PN: WO2004005342 LEQEPHE: 46 e itse protheine, Ipamorelin, NNC 26-0161
|
CAS |
170851-70-4
|
MF |
C38H49N9O5
|
MW |
711.853
|
Ponahalo |
Phofo e tšoeu
|
Kereiti |
Meriana ea Kereiti
|
Ho hloeka |
99%
|
Tšebeliso |
Hormone ea kholo ea sekhukhu e amohela mokelikeli o kopantseng liprotheine o tlamang ghrelin mme o bapala karolo ea matla a homeostasis le taolo ea boima ba 'mele.
|
Tlhaloso:
Ipamorelin ke se sibolloang se secha se hahang sa mesifa se fumanang tlhokomelo e ngata ho
lefats'e la ho haha 'mele. Ke peptide ea maiketsetso e nang le thepa e matla ea kholo ea kholo ea kholo. Mme thepa ena e lokollang GH ke eona e khahlang baatlelete le lihahi tsa 'mele kaha li ka etsa phapang e kholo ho bongata ba mesifa eo o ka e holang le hore na o chesa mafura kapele hakae.
Ipamorelin ke penta-peptide. (Aib-His-D-2-Nal-D- Phe-Lys-NH2) Hape, matla ao e a bonang a ka etsa hore Growth Hormon (GH) ea khale e felloe ke nako. re hlile re batla ho tseba hore na peptide ee e makatsang e khona ho e etsa, e sebelisoa joang, 'me e bapisoa joang le li-peptide tse ling tsa GHRP?
Baatlelete ba nka Ipamorelin ka litekanyo tsa 200mcg -300mcg, makhetlo a mabeli kapa a mararo ka letsatsi, ba sebelisa nale e nyane ea insulin ho e enta. Hangata ba qala ka lethal dose e tlase hobane litla-morao li ka kenyelletsa hlooho kapa se utloang eka ke ho potlaka ha hlooho. e nkuoe neng kapa neng empa e nka hoo e ka bang metsotso e 30-45 pele ho ikoetlisa ho ka utloahala ho lokile ka lebaka la pulse ea Growth Hormon (GH) eo e fanang ka eona e lumellang kholo e kholo.
Boithuto ka litlamorao tsa Ipamorelin mabapi le kholo ea masapo, boima ba 'mele, le tokollo ea GH li bonts'itse liqeto tse ling tse khahlisang. Ketsahalong e 'ngoe, ho ile ha fanoa ka litekanyetso tse fapaneng nakong ea matsatsi a 15 ho leka liketso tsa sehlopha.
Ho bile le phello e ikhethileng le e itšetlehileng ka tekanyetso ea boima ba 'mele leha ho le joalo, sehlopha sa kalafo ha sea ka sa bontša phetoho maemong ohle a IGF-I. Hape sehlopha sa kalafo ha sea ka sa hlahisa matšoao a serum
ntshetsopele. Mohlala, palo ea lisele tse karolong e pharaletseng ea tibia (shinbone) ha ea fetoha haholo. Hona ke ntho e ntle hobane e fana ka maikutlo a kholo ea mesifa e nang le menyetla e fokolang ea ho holofala ha masapo kapa lefufuru.
Karabelo ea pituitary ho iVDose e mabifi ea Ipamorelin e bonts'itse hore litekanyetso tsa plasma GH li fokotsehile haholo athe ha lia ka tsa fetoha kamora tekanyo e tšoanang ea GHRH. Sena ke ntho e ntle kaha se fana ka maikutlo a hore Ipamorelin e kanna ea se ke ea fokotsa tlhahiso ea 'mele ea tlhaho ea GH - hape e bonts'a hore Ipamorelin ke khetho ea GH e khethiloeng.
Ipamorelin ha e bake tlala e etsang hore e be molemo ho ba jang lijo tse thibetsoeng tsa khalori. Ho hlakile hore litlamorao tsa Ipamorelin lia ntlafatsoa ha li kopantsoe le li-anabolic steroids hobane le tsona li susumetsa tlhahiso le tlhahiso ea Growth Hormon / Insulin Growth Factor.
Tlhaloso ea IPamorelin
Litlhaloso
|
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Ponahalo |
Phofo e tšoeu
|
||||||
Ponahalo ea tharollo |
Tse sa bonahaleng
|
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Mmala oa tharollo |
Ha e na mmala
|
||||||
PH |
nyehelo
|
||||||
Phetoho e khethehileng ea Optical (c = 0.5,95% HAc) |
nyehelo
|
||||||
Ho hloeka (ke HPLC) |
≥98.00% ~ 99.90%
|
||||||
Litšila tsohle (ka HPLC) |
.002.00% ~ 0.05%
|
||||||
Ho se hloeke ho se nang molekane (ke HPLC) |
≤0.50% ~ 0.08%
|
||||||
Boitsebiso ba Metsi (Karl Fischer) |
.4.80%
|
||||||
Boitsebiso ba Acetate (ke HPLC) |
.6.80%
|
||||||
Boitsebiso ba Peptide (ka% N) |
≥88.00%
|
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Sebopeho sa Amino Acaid |
± 10% ea thuto
|
||||||
Thlahlobo (Ka anhydrous, acetic acid ntle) |
95.0% ~ 105.0%
|
||||||
Ho qhibiliha
|
nyehelo |
Litlaleho:
Ipamorelin (kapa NNC 26-0161) ke ea li-peptide tse laolang hobane ke GH e ntšang protheine; Moketane oa eona o mokhutšoanyane haholo mme o na le li-amino acid tse hlano feela. Boima ba eona ba limolek'hule ke 711.86 mme mokhoa oa eona oa limolek'hule ke C38H49N9O5. Ipamorelin e entsoe ka mokhoa o mocha oa ho etsisa ghrelin ka hona e na le bokhoni ba ho ntlafatsa motility ea ka mpeng. Ho na le liteko tse 'maloa tse ntseng li tsoela pele tsa kliniki le ipamorelin hajoale. Lithuto tsa pele tsa HGr-peptide ho kenyeletsoa NNC 26-0161 li qalile mathoasong a bo-1990. Hape setsi sena sa lipatlisiso ke sephiri se khethiloeng sa G-hormone le ghonlin receptor's agonist. Ha liprotheine tse ling ipamorelin e sebetsana le li-receptor tse kang tsa GHRP ho lokolla li-hormone tsa kholo ho tsoa tšoelesa ea pituitary. Empa ho fapana le li-peptide tse 'maloa tsa li-hormone mofuta ona oa pentapeptide ha o ntše molumo o tšoanang oa metsoako e joalo ka cortisol le acetylcholine, mme seo se e etsa mokhethoa ea khabane bakeng sa lipatlisiso tse tlang. Ntle le moo, NNC 26-0161 ke mofuta o tsitsitseng oa ghrelin mme o na le nako e telele ea bophelo, mme e baka tšusumetso ea bobeli ka ho etsa hore methapo ea kutlo e nyakalle.
Kopo:
Ipamorelin ke peptide e khahlisang e nkuoang 300mcg habeli ka letsatsi kapa u ka theola lethal dose makhetlo a 3 ka letsatsi, litla-morao ke ho potlaka ha hlooho, ke khothaletsa ho nka metsotso ena e 30 pele u ikoetlisa, ka gear, Ipamorelin ke pentapeptide e ncha le e matla ea maiketsetso e khethollang le thepa e ikhethileng ea "hormone" ea kholo (GH). Ka sepheo sa ho batlisisa litlamorao tsa sekhahla sa kholo ea masapo, boima ba 'mele le tokollo ea GH, Ipamorelin ka litekanyo tse fapaneng (0, 18, 90 le 450 μg / letsatsi) e ile ea entoa makhetlo a mararo ka letsatsi bakeng sa matsatsi a 15 ho leka lithuto,
Kamora ho ngoloa ha intraital Tetracycline ka matsatsi a 0, 6 le 13, LGR e ile ea khethoa ka ho lekanya sebaka se pakeng tsa lihlopha tse fapaneng tsa fluorescent ho metaphysis e haufi ea tibia. Ipamorelin e itšetlehileng ka tekanyetso ea LGD ho tloha ho 42 μm / ka letsatsi sehlopheng sa likoloi ho ea ho 44, 50, le 52 μm / ka letsatsi lihlopheng tsa kalafo. Ho ne ho boetse ho e-na le phello e boletsoeng le e itšetlehileng ka lethal dose ho nona ha 'mele. Kalafo ha ea ka ea ama maemo a IGF-I ka botlalo, kapa matšoao a serum a sebopeho sa masapo le ho hlaphoheloa ha 'mele.
Tlhahiso:
Haha mesifa e mosesane e thata, fokotsa mafura a 'mele le ho fokotsa ho boloka metsi le Ipamorelin ho tsoa Forever Young Medical Institute. E na le thuso bakeng sa: Lihahi tsa 'mele tse batlang ho tiisa; Batho ba tloaelehileng bakeng sa tahlehelo ea mafura le boleng bo ntlafalitsoeng ba mesifa; Batho ba baholo ba batla melemo e khahlanong le botsofali; Tlhabollo ea kotsi e potlakileng;
Melemo:
1. Khamphani ea rona ke feme e etellang pele ea tlhahiso ea China e sebakeng sa meriana sa lilemo tse ngata. Lisebelisoa tsa lihlahisoa tsa rona: US, UK, Canada, Australia, Brazil, Russia, Portugal, Latvia, Switzerland, Iceland, Ukraine, Jeremane, France, Netherlands, Belgium, Peru, Sweden, New Zealand, Czech Republic, Lithuania, Ireland , Tunisia, Mexico, Greece, Puerto Rico, Thailand, Israel joalo-joalo. Mokhoa oa ho patala: T / T, mokhatlo oa Bophirimela, Moneygram.
2. Sephutheloana se masene. Liaparo tsa ho paka tseo u ka li khethang ka nepo li ka khethoa ho tšela moetlo ka polokeho. Kapa haeba u na le tsela ea hau e nepahetseng, e kanna ea nahaneloa.
3. Boleng bo holimo. Boleng bo phahameng bo netefalitsoe, hang ha bothata bofe kapa bofe bo fumaneha, sephutheloana se ne se tla tlosoa
uena.
4.Ts'ireletso ea Ts'ireletso: Ho romelloa ka Express (FedEx, UPS, DHL, EMS), ka moea. Moetapele ea hloahloa ka ho fetesisa o tla buelloa bakeng sa hau.
5. Re na le setoko, ka hona re ka tsamaisa kapele kapele ka lona letsatsi leo re fumanang tefo ka lona.
6. Tšebeletso e futhumetseng ea kamora ho rekisa bakeng sa hau 24/7. Potso efe kapa efe ea potso ea hau e tla rarolloa ho ea pele hang ha ho fihla
khoneha.
7. Ho tla fanoa ka theolelo ha u etsa odara e kholo.
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